{"id":2414,"date":"2023-03-29T16:28:31","date_gmt":"2023-03-29T07:28:31","guid":{"rendered":"https:\/\/www.insilico.jp\/blog\/?p=2414"},"modified":"2023-04-11T10:35:43","modified_gmt":"2023-04-11T01:35:43","slug":"kishida_virtual_library_cgbvs","status":"publish","type":"post","link":"https:\/\/www.insilico.jp\/blog\/2023\/03\/29\/kishida_virtual_library_cgbvs\/","title":{"rendered":"\u30ad\u30b7\u30c0\u5316\u5b66\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea\u306eCGBVS\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0"},"content":{"rendered":"\n<h2 class=\"wp-block-heading\">\u306f\u3058\u3081\u306b<\/h2>\n\n\n\n<p><a href=\"http:\/\/www.kishida.co.jp\/product\/discovery\/k-lb.html\">\u30ad\u30b7\u30c0\u5316\u5b66\u3055\u3093\u304c\u63d0\u4f9b\u3057\u3066\u3044\u308b\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea<\/a>\u306e\u4e00\u90e8\u306e\u5316\u5408\u7269\u306b\u3064\u3044\u3066CGBVS\u6cd5\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u3092\u3084\u3063\u3066\u307f\u307e\u3057\u305f\u3002\u3053\u306e\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea\u30fc\u306f\u30ad\u30b7\u30c0\u5316\u5b66\u3055\u3093\u304c\u6271\u3063\u3066\u3044\u308b\u30d3\u30eb\u30c7\u30a3\u30f3\u30b0\u30d6\u30ed\u30c3\u30af\u3092\u7d44\u307f\u5408\u308f\u305b\u3066\u5408\u6210\u3067\u304d\u308b\u3082\u306e\u3067\u30012\u6210\u5206\u7cfb\u30683\u6210\u5206\u7cfb\u306e2\u7a2e\u985e\u304c\u3042\u308a\u307e\u3059\u30022\u6210\u5206\u7cfb\u306e\u65b9\u306f\u5316\u5408\u7269\u6570\u304c800\u4e07\u500b\u4ee5\u4e0a\u3068\u591a\u304f\u5408\u6210\u306e\u5de5\u7a0b\u6570\u3082\u5c0f\u3055\u304f\u6bd4\u8f03\u7684\u5b89\u4fa1\u3060\u305d\u3046\u3067\u3059\u30023\u6210\u5206\u7cfb\u306f2\u6210\u5206\u7cfb\u3088\u308a\u5de5\u7a0b\u6570\u304c\u5927\u304d\u304f\u306a\u308a\u4fa1\u683c\u3082\u9ad8\u304f\u306a\u308b\u304c\u3001\u7acb\u4f53\u7684\u3067\u9762\u767d\u3044\u5316\u5408\u7269\u304c\u591a\u3044\u3068\u306e\u3053\u3068\u3067\u3059\u3002\u7279\u306bPPI\u963b\u5bb3\u5264\u3092\u5fd7\u5411\u3057\u305f\u8a2d\u8a08\u306b\u306a\u3063\u3066\u3044\u308b\u3088\u3046\u3067\u3059\u3002\u3053\u3061\u3089\u306e3\u6210\u5206\u7cfb\u306e\u30d0\u30fc\u30c1\u30e3\u30eb\u5316\u5408\u7269\u6570\u304c32\u4e07\u500b\u7a0b\u5ea6\u3068\u3001CGBVS\u6cd5\u306b\u3068\u3063\u3066\u4e01\u5ea6\u3088\u304b\u3063\u305f\u306e\u3067\u8a08\u7b97\u3057\u3066\u307f\u307e\u3057\u305f\u3002<\/p>\n\n\n\n<p>CGBVS\u6cd5\u306b\u3064\u3044\u3066\u306f\u4ee5\u4e0b\u306e\u8ad6\u6587\u3092\u53c2\u7167\u3057\u3066\u304f\u3060\u3055\u3044\u3002<\/p>\n\n\n\n<ul class=\"wp-block-list\"><li><a href=\"https:\/\/doi.org\/10.1093\/bioinformatics\/btn162\">YABUUCHI, Hiroaki, et al. Analysis of multiple compound\u2013protein interactions reveals novel bioactive molecules. Molecular systems biology, 2011, 7.1: 472.<\/a><\/li><li><a href=\"https:\/\/doi.org\/10.3390\/molecules26175131\">KANAI, Chisato, et al. Computational Prediction of Compound\u2013Protein Interactions for Orphan Targets Using CGBVS. Molecules, 2021, 26.17: 5131.<\/a><\/li><\/ul>\n\n\n\n<p>CGBVS\u306e\u7279\u5fb4\u306e\u4e00\u3064\u306b\u8907\u6570\u30bf\u30f3\u30d1\u30af\u8cea\u306b\u5bfe\u3059\u308b\u5316\u5408\u7269\u306e\u7d50\u5408\u4e88\u6e2c\u3092\u4e00\u5ea6\u306b\u8a55\u4fa1\u3067\u304d\u308b\u3053\u3068\u304c\u3042\u308a\u307e\u3059\u3002\u73fe\u5728\u306fChEMBL30\u306e\u30c7\u30fc\u30bf\u3092\u57fa\u306b\u3057\u3066\u30e2\u30c7\u30eb\u3092\u4f5c\u6210\u3057\u3066\u304a\u308a\u30019\u7a2e\u985e\u306e\u30e2\u30c7\u30eb\u3067\u5408\u8a081595\u30bf\u30f3\u30d1\u30af\u8cea\u306b\u5bfe\u3057\u3066\u7d50\u5408\u4e88\u6e2c\u3059\u308b\u3053\u3068\u304c\u53ef\u80fd\u3067\u3059\u3002\u4eca\u56de\u306f3\u6210\u5206\u7cfb\u306e\u30d0\u30fc\u30c1\u30e3\u30eb\u5316\u5408\u726932\u4e07\u500b\u30921595\u30bf\u30f3\u30d1\u30af\u8cea\u306b\u5bfe\u3057\u3066\u7d50\u5408\u4e88\u6e2c\u30b9\u30b3\u30a2\u3092CGBVS\u6cd5\u306b\u3066\u8a55\u4fa1\u3057\u305f\u7d50\u679c\u3092\u7d39\u4ecb\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<h2 class=\"wp-block-heading\">\u8a08\u7b97\u65b9\u6cd5<\/h2>\n\n\n\n<p>CGBVS\u6cd5\u306f\u8a2d\u5b9a\u3055\u308c\u305f\u6d3b\u6027\u57fa\u6e96\u3067\u6d3b\u6027\u6709\u308a\u7121\u3057\u306e2\u30af\u30e9\u30b9\u306b\u30c7\u30fc\u30bf\u3092\u5206\u3051\u3066\u30012\u30af\u30e9\u30b9\u5206\u985e\u306e\u6a5f\u68b0\u5b66\u7fd2(SVM)\u3092\u5229\u7528\u3057\u3066\u6d3b\u6027\u4e88\u6e2c\u3059\u308b\u8a08\u7b97\u65b9\u6cd5\u3067\u3059\u3002\u8a73\u3057\u304f\u306f\u524d\u8ff0\u306e\u8ad6\u6587\u3092\u53c2\u7167\u3057\u3066\u304f\u3060\u3055\u3044\u3002<\/p>\n\n\n\n<p>\u8a08\u7b97\u5bfe\u8c61\u306f\u30ad\u30b7\u30c0\u5316\u5b66\u306e3\u6210\u5206\u7cfb\u306e\u30d0\u30fc\u30c1\u30e3\u30eb\u5316\u5408\u7269\u3067\u3001\u5316\u5408\u7269\u6570\u304c324,322\u500b\u3067\u3059\u3002\u8a08\u7b97\u65b9\u6cd5\u306f\u6211\u3005\u304c\u8ca9\u58f2\u3057\u3066\u3044\u308b\u30bd\u30d5\u30c8\u306eCzeekS\u3092\u5229\u7528\u3057\u3066\u3001\u4ee5\u4e0b\u306e9\u7a2e\u985e\u306e\u30e2\u30c7\u30eb\u3092\u5229\u7528\u3057\u30661595\u30bf\u30f3\u30d1\u30af\u8cea\u306b\u5bfe\u3057\u3066\u8a08\u7b97\u3092\u3057\u307e\u3057\u305f\u3002\u6d3b\u6027\u57fa\u6e96\u5024\u306f30uM\u3067\u3001IC50\u7b49\u304c30uM\u4ee5\u4e0b\u3067\u3042\u308c\u3070\u6d3b\u6027\u6709\u308a\u3068\u3057\u3066\u3044\u307e\u3059\u3002CGBVS\u306e\u30b9\u30b3\u30a2\u306f0\uff5e1\u307e\u3067\u306e\u5024\u3092\u53d6\u308a\u3001\u5316\u5408\u7269\u3068\u30bf\u30f3\u30d1\u30af\u8cea\u306e\u7d44\u307f\u5408\u308f\u305b\u304c\u6d3b\u6027\u3092\u6301\u3064\u78ba\u7387\u5024\u306e\u69d8\u306a\u610f\u5473\u3092\u6301\u3061\u307e\u3059\u3002\u6ce8\u610f\u3059\u3079\u304d\u306f\u30b9\u30b3\u30a2\u3068\u6d3b\u6027\u5024\uff08IC50\u7b49\uff09\u306b\u306f\u76f8\u95a2\u306f\u7121\u304f\u3001\u30b9\u30b3\u30a2\u304c1\u306b\u8fd1\u304f\u3066\u3082\u5fc5\u305a\u3057\u3082\u6d3b\u6027\u304c\u5f37\u3044\u3068\u4e88\u6e2c\u3057\u3066\u3044\u308b\u308f\u3051\u3067\u306f\u3042\u308a\u307e\u305b\u3093\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th class=\"has-text-align-left\" data-align=\"left\">\u30e2\u30c7\u30eb<\/th><th class=\"has-text-align-right\" data-align=\"right\">\u30bf\u30f3\u30d1\u30af\u8cea\u6570<\/th><th class=\"has-text-align-right\" data-align=\"right\">\u5b66\u7fd2\u30c7\u30fc\u30bf<\/th><\/tr><\/thead><tbody><tr><td class=\"has-text-align-left\" data-align=\"left\">Cytochrome P450<\/td><td class=\"has-text-align-right\" data-align=\"right\">39<\/td><td class=\"has-text-align-right\" data-align=\"right\">42,654<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">Esterase<\/td><td class=\"has-text-align-right\" data-align=\"right\">171<\/td><td class=\"has-text-align-right\" data-align=\"right\">106,874<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">GPCR<\/td><td class=\"has-text-align-right\" data-align=\"right\">259<\/td><td class=\"has-text-align-right\" data-align=\"right\">186,930<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">Ion channel<\/td><td class=\"has-text-align-right\" data-align=\"right\">180<\/td><td class=\"has-text-align-right\" data-align=\"right\">58,348<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">Kinase<\/td><td class=\"has-text-align-right\" data-align=\"right\">495<\/td><td class=\"has-text-align-right\" data-align=\"right\">200,000<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">Nuclear receptor<\/td><td class=\"has-text-align-right\" data-align=\"right\">42<\/td><td class=\"has-text-align-right\" data-align=\"right\">37,529<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">PPI<\/td><td class=\"has-text-align-right\" data-align=\"right\">53<\/td><td class=\"has-text-align-right\" data-align=\"right\">42,215<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">Protease<\/td><td class=\"has-text-align-right\" data-align=\"right\">235<\/td><td class=\"has-text-align-right\" data-align=\"right\">108,502<\/td><\/tr><tr><td class=\"has-text-align-left\" data-align=\"left\">Transporter<\/td><td class=\"has-text-align-right\" data-align=\"right\">121<\/td><td class=\"has-text-align-right\" data-align=\"right\">44,405<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h2 class=\"wp-block-heading\">CGBVS\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u7d50\u679c<\/h2>\n\n\n\n<p>\u5316\u5408\u7269\u304c\u7d0432\u4e07\u500b\u3067\u30bf\u30f3\u30d1\u30af\u8cea\u304c\u7d041600\u500b\u306a\u306e\u3067\u3001\u8a08\u7b97\u7d50\u679c\u306e\u30c7\u30fc\u30bf\u30dd\u30a4\u30f3\u30c8\u6570\u3068\u3057\u3066\u306f\u305d\u308c\u3089\u306e\u7a4d\u3067\u3042\u308b5.12\u5104\u7a0b\u3042\u308a\u307e\u3059\u3002\u30c7\u30fc\u30bf\u6570\u304c\u591a\u3059\u304e\u308b\u306e\u3067\u3001\u8a08\u7b97\u7d50\u679c\u306e\u5927\u307e\u304b\u306a\u69d8\u5b50\u3092\u78ba\u8a8d\u3059\u308b\u305f\u3081\u306b\u30d2\u30fc\u30c8\u30de\u30c3\u30d7\u306b\u307e\u3068\u3081\u3066\u307f\u307e\u3057\u305f\u3002\u5148\u305a\u306f\u30c7\u30fc\u30bf\u5168\u4f53\u306e\u69d8\u5b50\u306f\u4ee5\u4e0b\u306e\u56f3\u306e\u3088\u3046\u306b\u306a\u308a\u307e\u3057\u305f\u3002<\/p>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/All_Proteins-683x1024.png\" alt=\"\" class=\"wp-image-2418\" width=\"512\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/All_Proteins-683x1024.png 683w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/All_Proteins-200x300.png 200w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/All_Proteins-768x1152.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/All_Proteins-300x450.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/All_Proteins.png 800w\" sizes=\"auto, (max-width: 512px) 100vw, 512px\" \/><\/figure><\/div>\n\n\n\n<p>\u7e26\u8ef8\u306e\u5316\u5408\u7269\u306b\u3064\u3044\u3066\u306f32\u4e07\u500b\u3092k-means\u6cd5\u306b\u3088\u3063\u306650\u500b\u306e\u30af\u30e9\u30b9\u30bf\u30fc\u306b\u5206\u3051\u3066\u3044\u307e\u3059\u3002\u5316\u5408\u7269\u30b0\u30eb\u30fc\u30d7\u540d\u306fC0\uff5eC49\u307e\u3067\u3042\u308a\u307e\u3059\u3002\u6a2a\u8ef8\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u306b\u3064\u3044\u3066\u306f\u30e2\u30c7\u30eb\u6bce\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u3067\u307e\u3068\u3081\u3066\u3044\u307e\u3059\u3002\u5404\u5347\u76ee\u306e\u8272\u306f\u30b9\u30b3\u30a2\u306e\u5e73\u5747\u5024\u306b\u5fdc\u3058\u3066\u8272\u4ed8\u3051\u3057\u3066\u3044\u307e\u3059\u30023\u6210\u5206\u7cfb\u306e\u30ad\u30b7\u30c0\u5316\u5b66\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea\u30fc\u306fPPI\u963b\u5bb3\u5264\u3092\u5fd7\u5411\u3057\u305f\u8a2d\u8a08\u3068\u306e\u3053\u3068\u3067\u3059\u304c\u3001\u78ba\u304b\u306bPPI\u306b\u3064\u3044\u3066\u306f\u30b9\u30b3\u30a2\u304c\u9ad8\u3081\u306b\u51fa\u3066\u3044\u308b\u3088\u3046\u306b\u898b\u3048\u307e\u3059\u3002\u7279\u306bC48\u30b0\u30eb\u30fc\u30d7\u306e\u5316\u5408\u7269\u304cPPI\u963b\u5bb3\u5264\u306b\u826f\u3044\u3088\u3046\u306a\u6c17\u304c\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<p>\u3082\u3046\u5c11\u3057\u8a73\u3057\u304f\u30e2\u30c7\u30eb\uff08\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\uff09\u6bce\u306e\u30d2\u30fc\u30c8\u30de\u30c3\u30d7\u3092\u4ee5\u4e0b\u306b9\u7a2e\u985e\u793a\u3057\u3066\u3044\u304d\u307e\u3059\u3002\u7e26\u8ef8\u306f\u5316\u5408\u7269\u30b0\u30eb\u30fc\u30d7\uff08C0\uff5eC49\uff09\u3092\u793a\u3057\u3066\u3044\u3066\u3001\u6a2a\u8ef8\u306f\u30bf\u30f3\u30d1\u30af\u8cea\u3092\u30af\u30e9\u30b9\u30bf\u30ea\u30f3\u30b0\u3057\u305f\u3082\u306e\u3092\u793a\u3057\u3066\u304a\u308a\u307e\u3059\u3002\u30bf\u30f3\u30d1\u30af\u8cea\u306b\u3064\u3044\u3066\u3082k-means\u6cd5\u306b\u3088\u308a\u30af\u30e9\u30b9\u30bf\u30ea\u30f3\u30b0\u3057\u3066\u3044\u3066\u3001\u5404\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u6bce\u306b\u884c\u3044\u307e\u3057\u305f\u3002\u30af\u30e9\u30b9\u30bf\u30ea\u30f3\u30b0\u3057\u305f\u7d50\u679c\u3092\u30a8\u30af\u30bb\u30eb\u30d5\u30a1\u30a4\u30eb\u307e\u3068\u3081\u3066\u304a\u308a\u307e\u3059\u306e\u3067\u3001\u8a73\u3057\u304f\u306f\u3053\u3061\u3089\u306e\u30d5\u30a1\u30a4\u30eb\u3092\u53c2\u7167\u3057\u3066\u304f\u3060\u3055\u3044\u3002<\/p>\n\n\n\n<div class=\"wp-block-file\"><a id=\"wp-block-file--media-db2eb62b-a6e0-4d1e-bd43-97803673139c\" href=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/\u30af\u30e9\u30b9\u30bf\u30ea\u30f3\u30b0.xlsx\">\u30af\u30e9\u30b9\u30bf\u30ea\u30f3\u30b0<\/a><a href=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/\u30af\u30e9\u30b9\u30bf\u30ea\u30f3\u30b0.xlsx\" class=\"wp-block-file__button\" download aria-describedby=\"wp-block-file--media-db2eb62b-a6e0-4d1e-bd43-97803673139c\">\u30c0\u30a6\u30f3\u30ed\u30fc\u30c9<\/a><\/div>\n\n\n\n<h3 class=\"wp-block-heading\">Cytochrome P450 (CYP)<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP-853x1024.png\" alt=\"\" class=\"wp-image-2427\" width=\"640\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP-853x1024.png 853w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP-250x300.png 250w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP-768x922.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP-300x360.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP-850x1020.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/CYP.png 1000w\" sizes=\"auto, (max-width: 640px) 100vw, 640px\" \/><\/figure><\/div>\n\n\n\n<p>\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306eP1\u306b\u5bfe\u3057\u3066\u7279\u306b\u30b9\u30b3\u30a2\u304c\u9ad8\u3044\u50be\u5411\u304c\u3042\u308a\u307e\u3059\u3002P1\u306f\u5b9f\u306f\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u3067\u3001\u305d\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u306fCYP3A4\u3067\u3059\u3002\u3042\u3068\u4e3b\u3060\u3063\u305fCYP\u306b1A2, 2C9, 2C19, 2D6\u304c\u3042\u308a\u307e\u3059\u304c\u3001\u3053\u308c\u3089\u3082\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u3067\u3057\u305f\u3002\u4ee5\u4e0b\u306b\u307e\u3068\u3081\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P8<\/td><td>CYP1A2<\/td><\/tr><tr><td>P5<\/td><td>CYP2C9<\/td><\/tr><tr><td>P2<\/td><td>CYP2C19<\/td><\/tr><tr><td>P3<\/td><td>CYP2D6<\/td><\/tr><tr><td>P1<\/td><td>CYP3A4<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<p>\u3053\u306e\u56f3\u3092\u898b\u308b\u3068C17\u3084C16\u306b\u5c5e\u3059\u308b\u5316\u5408\u7269\u7fa4\u306fCYP\u306b\u5bfe\u3057\u3066\u30b9\u30b3\u30a2\u304c\u9ad8\u3044\u306e\u3067\u3001\u3053\u306e\u4e2d\u304b\u3089\u5316\u5408\u7269\u9078\u629e\u3059\u308b\u5834\u5408\u306f\u6ce8\u610f\u6df1\u304f\u898b\u308b\u5fc5\u8981\u304c\u3042\u308b\u304b\u3082\u3057\u308c\u307e\u305b\u3093\u3002<\/p>\n\n\n\n<h3 class=\"wp-block-heading\">Esterase<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase-853x1024.png\" alt=\"\" class=\"wp-image-2430\" width=\"640\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase-853x1024.png 853w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase-250x300.png 250w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase-768x922.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase-300x360.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase-850x1020.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Esterase.png 1000w\" sizes=\"auto, (max-width: 640px) 100vw, 640px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P3<\/td><td>Tyrosyl-DNA phosphodiesterase 1<\/td><\/tr><tr><td>P4<\/td><td>cAMP and cAMP-inhibited cGMP 3&#8242;,5&#8242;-cyclic phosphodiesterase 10A<\/td><\/tr><tr><td>P6<\/td><td>DNA-(apurinic or apyrimidinic site) endonuclease<\/td><\/tr><tr><td>P10<\/td><td>Ectonucleotide pyrophosphatase\/phosphodiesterase family member 2<\/td><\/tr><tr><td>P11<\/td><td>Monoglyceride lipase<\/td><\/tr><tr><td>P13<\/td><td>cAMP-specific 3&#8242;,5&#8242;-cyclic phosphodiesterase 4B<\/td><\/tr><tr><td>P17<\/td><td>Flap endonuclease 1<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h3 class=\"wp-block-heading\">GPCR<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-1024x1024.png\" alt=\"\" class=\"wp-image-2431\" width=\"768\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-1024x1024.png 1024w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-300x300.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-150x150.png 150w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-768x768.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-850x850.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR-45x45.png 45w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/GPCR.png 1200w\" sizes=\"auto, (max-width: 768px) 100vw, 768px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P10<\/td><td>Glucagon-like peptide 1 receptor<\/td><\/tr><tr><td>P11<\/td><td>Calcitonin gene-related peptide type 1 receptor<\/td><\/tr><tr><td>P22<\/td><td>C-C chemokine receptor type 2<\/td><\/tr><tr><td>P23<\/td><td>Neuropeptide S receptor<\/td><\/tr><tr><td>P25<\/td><td>C-X-C chemokine receptor type 3<\/td><\/tr><tr><td>P26<\/td><td>B1 bradykinin receptor<\/td><\/tr><tr><td>P3<\/td><td>C-C chemokine receptor type 5<\/td><\/tr><tr><td>P4<\/td><td>Melanin-concentrating hormone receptor 1<\/td><\/tr><tr><td>P7<\/td><td>Glucose-dependent insulinotropic receptor<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h3 class=\"wp-block-heading\">Ion channel<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch-853x1024.png\" alt=\"\" class=\"wp-image-2433\" width=\"640\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch-853x1024.png 853w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch-250x300.png 250w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch-768x922.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch-300x360.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch-850x1020.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Ionch.png 1000w\" sizes=\"auto, (max-width: 640px) 100vw, 640px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P1<\/td><td>P2X purinoceptor 7<\/td><\/tr><tr><td>P10<\/td><td>5-hydroxytryptamine receptor 3A<\/td><\/tr><tr><td>P12<\/td><td>P2X purinoceptor 3<\/td><\/tr><tr><td>P16<\/td><td>Cystic fibrosis transmembrane conductance regulator<\/td><\/tr><tr><td>P17<\/td><td>Voltage-dependent N-type calcium channel subunit alpha-1B<\/td><\/tr><tr><td>P2<\/td><td>Potassium voltage-gated channel subfamily H member 2 (hERG)<\/td><\/tr><tr><td>P4<\/td><td>Transient receptor potential cation channel subfamily V member 4<\/td><\/tr><tr><td>P5<\/td><td>Voltage-dependent T-type calcium channel subunit alpha-1H<\/td><\/tr><tr><td>P6<\/td><td>Sodium channel protein type 9 subunit alpha<\/td><\/tr><tr><td>P7<\/td><td>Voltage-dependent T-type calcium channel subunit alpha-1G<\/td><\/tr><tr><td>P9<\/td><td>Transient receptor potential cation channel subfamily V member 1<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<p>\u3053\u306e\u56f3\u3092\u898b\u308b\u3068C17\u306b\u5c5e\u3059\u308b\u5316\u5408\u7269\u7fa4\u306fP2\u30b0\u30eb\u30fc\u30d7(hERG)\u306b\u5bfe\u3057\u3066\u30b9\u30b3\u30a2\u304c\u9ad8\u3044\u306e\u3067\u3001<br>\u3053\u306e\u4e2d\u304b\u3089\u5316\u5408\u7269\u9078\u629e\u3059\u308b\u5834\u5408\u306fCYP\u3068\u540c\u69d8\u306b\u6ce8\u610f\u6df1\u304f\u898b\u308b\u5fc5\u8981\u304c\u3042\u308b\u304b\u3082\u3057\u308c\u307e\u305b\u3093\u3002<\/p>\n\n\n\n<h3 class=\"wp-block-heading\">Kinase<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Kinase-1024x878.png\" alt=\"\" class=\"wp-image-2434\" width=\"768\" height=\"659\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Kinase-1024x878.png 1024w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Kinase-300x257.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Kinase-768x658.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Kinase-850x729.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Kinase.png 1400w\" sizes=\"auto, (max-width: 768px) 100vw, 768px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P10<\/td><td>Serine\/threonine-protein kinase mTOR<\/td><\/tr><tr><td>P13<\/td><td>Mitogen-activated protein kinase 1<\/td><\/tr><tr><td>P19<\/td><td>Insulin-like growth factor 1 receptor<\/td><\/tr><tr><td>P21<\/td><td>Non-receptor tyrosine-protein kinase TYK2<\/td><\/tr><tr><td>P23<\/td><td>Mast\/stem cell growth factor receptor Kit<\/td><\/tr><tr><td>P26<\/td><td>Mitogen-activated protein kinase 14<\/td><\/tr><tr><td>P3<\/td><td>High affinity nerve growth factor receptor<\/td><\/tr><tr><td>P31<\/td><td>Mitogen-activated protein kinase 3<\/td><\/tr><tr><td>P32<\/td><td>Insulin receptor<\/td><\/tr><tr><td>P33<\/td><td>Tyrosine-protein kinase BTK<\/td><\/tr><tr><td>P38<\/td><td>Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform<\/td><\/tr><tr><td>P39<\/td><td>Epidermal growth factor receptor<\/td><\/tr><tr><td>P4<\/td><td>Mitogen-activated protein kinase 11<\/td><\/tr><tr><td>P41<\/td><td>Macrophage colony-stimulating factor 1 receptor<\/td><\/tr><tr><td>P42<\/td><td>Hexokinase-4<\/td><\/tr><tr><td>P43<\/td><td>ALK tyrosine kinase receptor<\/td><\/tr><tr><td>P44<\/td><td>Dual specificity protein kinase TTK<\/td><\/tr><tr><td>P45<\/td><td>Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform<\/td><\/tr><tr><td>P49<\/td><td>Cyclin-dependent kinase 9<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h3 class=\"wp-block-heading\">Nuclear receptor<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor-853x1024.png\" alt=\"\" class=\"wp-image-2435\" width=\"640\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor-853x1024.png 853w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor-250x300.png 250w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor-768x922.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor-300x360.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor-850x1020.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Nuclear_Receptor.png 1000w\" sizes=\"auto, (max-width: 640px) 100vw, 640px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P2<\/td><td>Nuclear receptor ROR-gamma<\/td><\/tr><tr><td>P3<\/td><td>Bile acid receptor<\/td><\/tr><tr><td>P7<\/td><td>Thyroid hormone receptor beta<\/td><\/tr><tr><td>P9<\/td><td>Glucocorticoid receptor<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h3 class=\"wp-block-heading\">PPI<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI-853x1024.png\" alt=\"\" class=\"wp-image-2436\" width=\"640\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI-853x1024.png 853w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI-250x300.png 250w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI-768x922.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI-300x360.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI-850x1020.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/PPI.png 1000w\" sizes=\"auto, (max-width: 640px) 100vw, 640px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P4<\/td><td>E3 ubiquitin-protein ligase Mdm2<\/td><\/tr><tr><td>P5<\/td><td>Bromodomain-containing protein 4<\/td><\/tr><tr><td>P7<\/td><td>Menin<\/td><\/tr><tr><td>P8<\/td><td>Apoptosis regulator Bcl-2<\/td><\/tr><tr><td>P9<\/td><td>E3 ubiquitin-protein ligase XIAP<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h3 class=\"wp-block-heading\">Protease<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-1024x1024.png\" alt=\"\" class=\"wp-image-2437\" width=\"768\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-1024x1024.png 1024w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-300x300.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-150x150.png 150w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-768x768.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-850x850.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease-45x45.png 45w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Protease.png 1200w\" sizes=\"auto, (max-width: 768px) 100vw, 768px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P10<\/td><td>Ubiquitin carboxyl-terminal hydrolase 2<\/td><\/tr><tr><td>P11<\/td><td>Renin<\/td><\/tr><tr><td>P12<\/td><td>Cathepsin S<\/td><\/tr><tr><td>P13<\/td><td>Prothrombin<\/td><\/tr><tr><td>P14<\/td><td>Coagulation factor XI<\/td><\/tr><tr><td>P15<\/td><td>Ubiquitin carboxyl-terminal hydrolase 1<\/td><\/tr><tr><td>P19<\/td><td>Cathepsin K<\/td><\/tr><tr><td>P20<\/td><td>Lysosomal Pro-X carboxypeptidase<\/td><\/tr><tr><td>P21<\/td><td>Beta-secretase 2<\/td><\/tr><tr><td>P22<\/td><td>Cathepsin D<\/td><\/tr><tr><td>P24<\/td><td>Neutrophil elastase<\/td><\/tr><tr><td>P25<\/td><td>Dipeptidyl peptidase 4<\/td><\/tr><tr><td>P28<\/td><td>Proprotein convertase subtilisin\/kexin type 9<\/td><\/tr><tr><td>P29<\/td><td>Complement factor D<\/td><\/tr><tr><td>P3<\/td><td>Coagulation factor X<\/td><\/tr><tr><td>P5<\/td><td>Beta-secretase 1<\/td><\/tr><tr><td>P9<\/td><td>Cathepsin B<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h3 class=\"wp-block-heading\">Transporter<\/h3>\n\n\n\n<div class=\"wp-block-image is-style-default\"><figure class=\"aligncenter size-large is-resized\"><img loading=\"lazy\" decoding=\"async\" src=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter-853x1024.png\" alt=\"\" class=\"wp-image-2438\" width=\"640\" height=\"768\" srcset=\"https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter-853x1024.png 853w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter-250x300.png 250w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter-768x922.png 768w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter-300x360.png 300w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter-850x1020.png 850w, https:\/\/www.insilico.jp\/blog\/wp-content\/uploads\/2023\/03\/Transporter.png 1000w\" sizes=\"auto, (max-width: 640px) 100vw, 640px\" \/><\/figure><\/div>\n\n\n\n<p>\u30b7\u30f3\u30b0\u30eb\u30c8\u30f3\u306e\u30bf\u30f3\u30d1\u30af\u8cea\u30b0\u30eb\u30fc\u30d7\u306e\u307f\u4ee5\u4e0b\u306e\u8868\u306b\u793a\u3057\u307e\u3059\u3002<\/p>\n\n\n\n<figure class=\"wp-block-table aligncenter is-style-stripes\"><table><thead><tr><th>\u30b0\u30eb\u30fc\u30d7<\/th><th>\u30bf\u30f3\u30d1\u30af\u8cea<\/th><\/tr><\/thead><tbody><tr><td>P1<\/td><td>Sodium-dependent serotonin transporter<\/td><\/tr><tr><td>P5<\/td><td>Sodium- and chloride-dependent glycine transporter 1<\/td><\/tr><tr><td>P7<\/td><td>ATP-dependent translocase ABCB1<\/td><\/tr><tr><td>P8<\/td><td>Solute carrier family 2, facilitated glucose transporter member 1<\/td><\/tr><\/tbody><\/table><\/figure>\n\n\n\n<h2 class=\"wp-block-heading\">\u7d50\u679c\u30d5\u30a1\u30a4\u30eb<\/h2>\n\n\n\n<p>\u3053\u306e\u30d6\u30ed\u30b0\u3067\u8a08\u7b97\u3057\u305f\u7d50\u679c\uff08\u751f\u30c7\u30fc\u30bf\uff09\u3092\u4ee5\u4e0b\u306e\u30ea\u30f3\u30af\u304b\u3089\u30c0\u30a6\u30f3\u30ed\u30fc\u30c9\u3067\u304d\u307e\u3059\u3002\u69cb\u9020\u5f0f\u30c7\u30fc\u30bf\u306b\u3064\u3044\u3066\u306f<a href=\"https:\/\/www.kishida.co.jp\/inquiry\/input\">\u30ad\u30b7\u30c0\u5316\u5b66\u306e\u65b9\u3078\u554f\u3044\u5408\u308f\u305b<\/a>\u9802\u3051\u308c\u3070\u5165\u624b\u3067\u304d\u307e\u3059\u3002\u3053\u308c\u3089\u306e\u30c7\u30fc\u30bf\u3092CGBVS\u6cd5\u3084\u30ad\u30b7\u30c0\u5316\u5b66\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea\u306e\u8a55\u4fa1\u306a\u3069\u306b\u3054\u5229\u7528\u9802\u3051\u308b\u3068\u5e78\u3044\u3067\u3059\u3002<\/p>\n\n\n\n<p><a href=\"https:\/\/drive.google.com\/uc?export=download&amp;id=1xP5e-luDaoO2HfTs-f9sxBY1DRij5vs2\" target=\"_blank\" rel=\"noreferrer noopener\">Raw Data<\/a><\/p>\n\n\n\n<p>Raw Data \u306b\u542b\u307e\u308c\u308b\u30d5\u30a1\u30a4\u30eb\u306b\u3064\u3044\u3066<\/p>\n\n\n\n<table id=\"tablepress-5\" class=\"tablepress tablepress-id-5\">\n<thead>\n<tr class=\"row-1\">\n\t<th class=\"column-1\">\u30d5\u30a1\u30a4\u30eb\u540d<\/th><th class=\"column-2\">\u30d5\u30a1\u30a4\u30eb\u306e\u5185\u5bb9<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr class=\"row-2\">\n\t<td class=\"column-1\">cyp_out_all.txt<\/td><td class=\"column-2\">Cytochrome\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-3\">\n\t<td class=\"column-1\">esterase_out_all.txt<\/td><td class=\"column-2\">Esterase\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-4\">\n\t<td class=\"column-1\">gpcr_out_all.txt<\/td><td class=\"column-2\">GPCR\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-5\">\n\t<td class=\"column-1\">ionch_out_all.txt<\/td><td class=\"column-2\">Ion channel\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-6\">\n\t<td class=\"column-1\">kinase_out_all.txt<\/td><td class=\"column-2\">Kinase\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-7\">\n\t<td class=\"column-1\">nhr_out_all.txt<\/td><td class=\"column-2\">Nuclear receptor\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-8\">\n\t<td class=\"column-1\">ppi_out_all.txt<\/td><td class=\"column-2\">PPI\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-9\">\n\t<td class=\"column-1\">protease_out_all.txt<\/td><td class=\"column-2\">Protease\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-10\">\n\t<td class=\"column-1\">trans_out_all.txt<\/td><td class=\"column-2\">Transporter\u6a19\u7684\u30bf\u30f3\u30d1\u30af\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u30c7\u30fc\u30bf<\/td>\n<\/tr>\n<tr class=\"row-11\">\n\t<td class=\"column-1\">CompoundClusterLabels.csv<\/td><td class=\"column-2\">\u5316\u5408\u7269ID\u3068\u30af\u30e9\u30b9\u30bf\u30fc\u30e9\u30d9\u30eb\u306eCSV\u30d5\u30a1\u30a4\u30eb<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<!-- #tablepress-5 from cache -->","protected":false},"excerpt":{"rendered":"<p>\u306f\u3058\u3081\u306b \u30ad\u30b7\u30c0\u5316\u5b66\u3055\u3093\u304c\u63d0\u4f9b\u3057\u3066\u3044\u308b\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea\u306e\u4e00\u90e8\u306e\u5316\u5408\u7269\u306b\u3064\u3044\u3066CGBVS\u6cd5\u306b\u3088\u308b\u30d7\u30ed\u30d5\u30a1\u30a4\u30ea\u30f3\u30b0\u3092\u3084\u3063\u3066\u307f\u307e\u3057\u305f\u3002\u3053\u306e\u30d0\u30fc\u30c1\u30e3\u30eb\u30e9\u30a4\u30d6\u30e9\u30ea\u30fc\u306f\u30ad\u30b7\u30c0\u5316\u5b66\u3055\u3093\u304c\u6271\u3063\u3066\u3044\u308b\u30d3\u30eb\u30c7\u30a3\u30f3\u30b0\u30d6\u30ed\u30c3\u30af\u3092\u7d44\u307f\u5408\u308f\u305b\u3066&#8230;<\/p>\n","protected":false},"author":5,"featured_media":0,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[118,4],"tags":[],"class_list":["post-2414","post","type-post","status-publish","format-standard","hentry","category-ai-drug-discovery","category-cgbvs-czeeks"],"yoast_head":"<!-- This site is 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